Quick Guide to Uncommon Stimulants

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2-MDP - Dissociative anaesthetic, NMDA antagonist, simlar effects to PCP in animals, (-) isomer is active. Roughly 1/3rd

potency of amphetamine by weight. Lasts over 24 hours.

2C-B-BZP - Benzylpiperazine base with ring-sub pattern of 2c-b. Not a phenethylamine, doesn't produce psychedelic effects.

Lasts 3-6 hours. Was sold in Japan in "smartshops"

A-366/833 - Agonist at neural nicotinic acetylcholine receptors selective for α4β2 subtype. Been researched as an analgesic.

Hasn't passed clinical trials.

A-84/543 ^ That and is used as the "standard" for this family of compounds.

2-Acetoxycocaine - Quicker onset than Cocaine. Four fold increase over cocaine in binding potency for dopamine. And 35 fold

enhanced affinity for the norepinephrine. Reduced selectivity for serotonin. Interesting structure.

Adrafinil - Prodrug of Modafinil, unregulated in the US. 1 hour half life.

AL-1095 - Centrally acting, comparable efffects to amp. developed by Bristol in the 70's.

Altinicline (SIB-1508Y) agonist at neural nicotinic acetylcholine receptors similar to A-366. Releases Dopamine and

Acetylcholine in both rodent and primate models. Progressed into Phase 2 clinical trials for Parkinson's.

Amfepramone - Diethylcathinone. By itself lacks any affinity for monoamine transporters and functions as a prodrug to ethcathinone. Very weak dopaminergic and serotonergic. 10-20x stronger on norepinephrine in comparison. Basically can be considered NRA's. Is currently Schedule IV in the United States. Class C drug in the UK. Apparently known as "tombstones" in the UK.