Uncommon Benzodiazepines: Difference between revisions
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(1,4-Benzodiazepines) |
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:Debazepide - (MK-329) Lacking affinity for GABA-A, instead acting as a Cholecystokinin antagonist selective for the CCK-A subtype Appetite stimulanting. | :Debazepide - (MK-329) Lacking affinity for GABA-A, instead acting as a Cholecystokinin antagonist selective for the CCK-A subtype Appetite stimulanting. | ||
:Diclazepam - RC. Meta's into 6-chloro-temazepam/delorazepam/desmethyldiazepam.Actually name: Chlorodiazepam | :Diclazepam - RC. Meta's into 6-chloro-temazepam/delorazepam/desmethyldiazepam. Actually name: Chlorodiazepam | ||
:Doxefazepam - Used therapeutically as a hypnotic. 2-4x more potent than Dalmane/Flurazepam. | :Doxefazepam - Used therapeutically as a hypnotic. 2-4x more potent than Dalmane/Flurazepam. | ||
:Ethyl Carfluzepate - Similar to Ethyl Loflazepate | :Ethyl Carfluzepate - Similar to Ethyl Loflazepate, Mainly Sedative/Hypnotic. | ||
:Ethyl Dirazepate - Anxiolytic/Hypnotic. Uninteresting. | :Ethyl Dirazepate - Anxiolytic/Hypnotic. Uninteresting. | ||
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:Flubromazepam - (RC) 8mg = 10mg diazepam. | :Flubromazepam - (RC) 8mg = 10mg diazepam. | ||
:Fletazepam - More muscle relaxant (GABA-B?) Most closely related to Halazepam and Quazepam. | :Fletazepam - More muscle relaxant (GABA-B?) Most closely related to Halazepam and Quazepam. | ||
:Fludiazepam - Maeketed in Taiwan/Japan in .25mg tablets (Erispan) 4 times more binding affinity towards GABA then Diazepam. Interesting. | :Fludiazepam - Maeketed in Taiwan/Japan in .25mg tablets (Erispan) 4 times more binding affinity towards GABA then Diazepam. Interesting. | ||
Revision as of 08:50, 28 October 2013
1,4-Benzodiazepines
- Camazepam - Dimethyl Carbamate (Gaba-B?) ester of Temazepam. Has little anticonvulsant/hypnotic/relaxant properties. Very low affinity for all Benzo receptors. Meta. into Temazepam. Is believed to increase attention(?) High oral BA (90%)(A.K.A Albego, Limpidon, and Paxor) Was scripted in Italy/Spain/Switzerland. 6-11 hour Half life.
- Elfazepam - Appetite stimulanting (Like antipyschs?) Sedative/Anxiolytic. Interesting and the stem of one of my names!
- Carburazepam - Could be an analogue of Temazepam/Camazepam. Will research further
- Cinolazepam - Has all the normal benzo properties. Has strong sedative properties, used primarily used as an hypnotic... Interesting. Will look further into possible analogues.
- Cyprazepam - Once again, nothing on it. Sedative-hypnotic... Will look further into possible analogues.
- Delorazepam - (Chlordesmethyldiazepam) Deriv. of Desmethyldiazepam. Marketed in Italy, available under EN and Dadumir. Active metabolite of Diclazepam and Cloxazolam. Mainly used as an anxiolytic because of long half life (80-115 hours) BA is around 77%. Peak plasma is within an hour. 1mg=10mg diazepam.
- Demoxepam - Metabolite of Chloridiazepoxide (Librium) Uninteresting. 35-40 hour half life.
- Debazepide - (MK-329) Lacking affinity for GABA-A, instead acting as a Cholecystokinin antagonist selective for the CCK-A subtype Appetite stimulanting.
- Diclazepam - RC. Meta's into 6-chloro-temazepam/delorazepam/desmethyldiazepam. Actually name: Chlorodiazepam
- Doxefazepam - Used therapeutically as a hypnotic. 2-4x more potent than Dalmane/Flurazepam.
- Ethyl Carfluzepate - Similar to Ethyl Loflazepate, Mainly Sedative/Hypnotic.
- Ethyl Dirazepate - Anxiolytic/Hypnotic. Uninteresting.
- Ethyl Loflazepate - Normal Benzo effects. Problems with very high doses (What doses?) Half life is 51-103 hours. Scripted in Mexico (Victan). Seems... really toxic at all doses.
- Flubromazepam - (RC) 8mg = 10mg diazepam.
- Fletazepam - More muscle relaxant (GABA-B?) Most closely related to Halazepam and Quazepam.
- Fludiazepam - Maeketed in Taiwan/Japan in .25mg tablets (Erispan) 4 times more binding affinity towards GABA then Diazepam. Interesting.