Quick Guide to Uncommon Stimulants: Difference between revisions

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2-MDP - Dissociative anaesthetic, NMDA antagonist, simlar effects to PCP in animals, (-) isomer is active. Roughly 1/3rd potency of amphetamine by weight. Lasts over 24 hours.  
:2-MDP - Dissociative anaesthetic, NMDA antagonist, simlar effects to PCP in animals, (-) isomer is active. Roughly 1/3rd potency of amphetamine by weight. Lasts over 24 hours.  


2C-B-BZP - Benzylpiperazine base with ring-sub pattern of 2c-b. Not a phenethylamine, doesn't produce psychedelic effects. Lasts 3-6 hours. Was sold in Japan in "smartshops"  
:2C-B-BZP - Benzylpiperazine base with ring-sub pattern of 2c-b. Not a phenethylamine, doesn't produce psychedelic effects. Lasts 3-6 hours. Was sold in Japan in "smartshops"  


A-366/833 - Agonist at neural nicotinic acetylcholine receptors selective for α4β2 subtype. Been researched as an analgesic. Hasn't passed clinical trials.  
:A-366/833 - Agonist at neural nicotinic acetylcholine receptors selective for α4β2 subtype. Been researched as an analgesic. Hasn't passed clinical trials.  


A-84/543 ^ That and is used as the "standard" for this family of compounds.  
:A-84/543 ^ That and is used as the "standard" for this family of compounds.  


2-Acetoxycocaine - Quicker onset than Cocaine. Four fold increase over cocaine in binding potency for dopamine. And 35 fold enhanced affinity for the norepinephrine. Reduced selectivity for serotonin. Interesting structure.  
:2-Acetoxycocaine - Quicker onset than Cocaine. Four fold increase over cocaine in binding potency for dopamine. And 35 fold enhanced affinity for the norepinephrine. Reduced selectivity for serotonin. Interesting structure.  


Adrafinil - Prodrug of Modafinil, unregulated in the US. 1 hour half life.  
:Adrafinil - Prodrug of Modafinil, unregulated in the US. 1 hour half life.  


AL-1095 - Centrally acting, comparable efffects to amp. developed by Bristol in the 70's.  
:AL-1095 - Centrally acting, comparable effects to amp. developed by Bristol in the 70's.  


Altinicline (SIB-1508Y) agonist at neural nicotinic acetylcholine receptors similar to A-366. Releases Dopamine and Acetylcholine in both rodent and primate models. Progressed into Phase 2 clinical trials for Parkinson's.
:Altinicline (SIB-1508Y) agonist at neural nicotinic acetylcholine receptors similar to A-366. Releases Dopamine and Acetylcholine in both rodent and primate models. Progressed into Phase 2 clinical trials for Parkinson's.


Amfepramone - Diethylcathinone. By itself lacks any affinity for monoamine transporters and functions as a prodrug to ethcathinone. Very weak dopaminergic and serotonergic. 10-20x stronger on norepinephrine in comparison. Basically can be considered NRA's. Is currently Schedule IV in the United States. Class C drug in the UK. Apparently known as "tombstones" in the UK.  
:Amfepramone - Diethylcathinone. By itself lacks any affinity for monoamine transporters and functions as a prodrug to ethcathinone. Very weak dopaminergic and serotonergic. 10-20x stronger on norepinephrine in comparison. Basically can be considered NRA's. Is currently Schedule IV in the United States. Class C drug in the UK. Apparently known as "tombstones" in the UK.  


2-amino-1,2-dihydronaphthalene - Also known as 2-AD, rigid analogue of phenylisobutylamine and substitutes amphetamine for it in rat discrimination tests, 1/4th the potency. Closely related to 2-aminotetralin.  
:2-amino-1,2-dihydronaphthalene - Also known as 2-AD, rigid analogue of phenylisobutylamine and substitutes amphetamine for it in rat discrimination tests, 1/4th the potency. Closely related to 2-aminotetralin.  


2-Aminoindane - 2-AI(RC) Psychoactive compound. Rigid analogue of amphetamine.  
:2-Aminoindane - 2-AI(RC) Psychoactive compound. Rigid analogue of amphetamine.  


5-(2-aminopropyl)indole - 5-IT(RC) indole derivative. Preparation was first reported in 1962 by Albert Hofmann. Positional isomer of AMT. Closer chemically resembles  
:5-(2-aminopropyl)indole - 5-IT(RC) indole derivative. Preparation was first reported in 1962 by Albert Hofmann. Positional isomer of AMT. Closer chemically resembles Phethylamines like 5-apb and the likes. Falls under the Analog act in the US with AMT.


Phethylamines like 5-apb and the likes. Falls under the Analog act in the US with AMT.  
:6-(2-Aminopropyl)indole - ^. But it has been shown to increase hemoglobin levels in the bloodstream.  


6-(2-Aminopropyl)indole - ^. But it has been shown to increase hemoglobin levels in the bloodstream.  
:Aminorex - Known by many other names. Anorectic stimulant. Is classed within the 2-amino-5-aryl oxazoline class. Closely related to 4-methylaminorex. Shown to have locomotor stimulant effects, lying midway between dextro-amp and Meth. Attributed to the release of cathecholamines. Retired from the market after it was found to result in pulmonary hypertension.  


Aminorex - Known by many other names. Anorectic stimulant. Is classed within the 2-amino-5-aryl oxazoline class. Closely related to 4-methylaminorex. Shown to have locomotor stimulant effects, lying midway between dextro-amp and Meth. Attributed to the release of cathecholamines. Retired from the market after it was found to result in pulmonary hypertension.  
:2-Aminotetralin - (2-AT) consiting of a tetralin group combined with an anime. Rigid analogue of phenylisobutylamine. Fully substitutes for D-Amp in rat discrimination tests. Although at 1/8th the potency. Inhibits the reuptake of serotonin and norepinephrine. Likely induces their release as well. Also likely to act of Dopamine on account of the D-Amp.  


2-Aminotetralin - (2-AT) consiting of a tetralin group combined with an anime. Rigid analogue of phenylisobutylamine. Fully substitutes for D-Amp in rat discrimination tests.  
:Amiphenazole - Traditionally used as an antidote for Barb/opioid overdose. Mixed with bemegride. As well as poisoning from other depressants.  


Although at 1/8th the potenct. Inhibits the reuptake of serotonin and norepinephrine. Likely induces their release as well. Also likely to act of Dopamine on account of the D-Amp.
:Ampyzine - Pyrazine derivative. That's all I could find with my limited research.
 
:AR-R17779 - Drug that acts as a potent and selective full agonist for the α7 subtype of neural nicotinic acetylcholine receptors. Nootropic effects in animal sudies.
 
:Armodafinal - Basically like all other versions of the ***final's nothing popped very interesting.
 
:Bemegride - Used in barb overdoses. "Popularized" by The suspected Serial Killer Dr. John Bodkin Adams.
 
:Benocyclidine - (BCP/BTCP) RC of the arylcyclohexylamine class. Acts as a Potent and Selective DRI. Pure DRI with negligible affintity for NMDA. Lacks every other propeties in effects, minus stimulant. Found in several MDMA presses.
 
:3-benzhydrylmorpholine - Developed in the 50's by American Home Products Corp. Stimulant and anoretctic effects. Related to pipradrol and phenmetrazine.
 
:Benzofuranylpropylaminopentance - ((-)-BPAP) Catecholaminergic and Serotonergic activity enhancer. Only increases the amount of neurotransmitters that get released. Weak MAO-A inhibitor. Showen to have neuroprotective effects similar to selegiling.  
 
:Benzooylthiomethylecgonine - Cocaine Analogue which has a sulfur in place of an oxygen on the single bonded benzoyl ester. Thus lowering potency.
 
:1-Benzyl-4-(2-(diphenylmethoxy)ethyl)piperidine - Acts as a potent and selective DRI.
 
:Benzylpipeazine - BZP, that's about it. 
 
:2-benzylpipeazine - 20x less potent than MPH and desoxypipadrol. Synthetic intermediate in other drugs :o. Boring stuff.
 
:4-benzylpipeazine - The exact opposite of ^^. Acts as a MAOI with 20 to 48 fold selectivity for releasing dopamine versus serotonin.
 
:Brasofensine - Phehyltropane. Effective in stimulating LMA and reversing akinesia. Idunknow.   
 
:Bromantane - Stimulant with anxiolytic properties developed in Russia during the late 1980's. DSRI. Has an anticholinergic effect at very high doses. Used as a doping agent for athletic performance. No withdrawal symptoms!
 
:BTS 74,398 - Weird structure, centrally acting stimulant drug. Acts as a triple reuptake inhibitor.  
 
:Butylolylquinuclidine - Was made to replace cocaine in cocaine addiction, while longest lasting and less potent.
 
:Camfetamine - N-Methyl homologue of fencamfamine. Apparently replaced mephedrone after it's banning?
 
:Meta-Chlorophenylpiperazine
 
:Cilboamine - NDRI, has stimulant and anti-dep effects.
 
:Clofeniciclan - Dopamine-releasing agent developed in the 50's. Proved unpopular as a treatment because of its pronounced stimulant activity

Latest revision as of 21:18, 3 February 2014

2-MDP - Dissociative anaesthetic, NMDA antagonist, simlar effects to PCP in animals, (-) isomer is active. Roughly 1/3rd potency of amphetamine by weight. Lasts over 24 hours.
2C-B-BZP - Benzylpiperazine base with ring-sub pattern of 2c-b. Not a phenethylamine, doesn't produce psychedelic effects. Lasts 3-6 hours. Was sold in Japan in "smartshops"
A-366/833 - Agonist at neural nicotinic acetylcholine receptors selective for α4β2 subtype. Been researched as an analgesic. Hasn't passed clinical trials.
A-84/543 ^ That and is used as the "standard" for this family of compounds.
2-Acetoxycocaine - Quicker onset than Cocaine. Four fold increase over cocaine in binding potency for dopamine. And 35 fold enhanced affinity for the norepinephrine. Reduced selectivity for serotonin. Interesting structure.
Adrafinil - Prodrug of Modafinil, unregulated in the US. 1 hour half life.
AL-1095 - Centrally acting, comparable effects to amp. developed by Bristol in the 70's.
Altinicline (SIB-1508Y) agonist at neural nicotinic acetylcholine receptors similar to A-366. Releases Dopamine and Acetylcholine in both rodent and primate models. Progressed into Phase 2 clinical trials for Parkinson's.
Amfepramone - Diethylcathinone. By itself lacks any affinity for monoamine transporters and functions as a prodrug to ethcathinone. Very weak dopaminergic and serotonergic. 10-20x stronger on norepinephrine in comparison. Basically can be considered NRA's. Is currently Schedule IV in the United States. Class C drug in the UK. Apparently known as "tombstones" in the UK.
2-amino-1,2-dihydronaphthalene - Also known as 2-AD, rigid analogue of phenylisobutylamine and substitutes amphetamine for it in rat discrimination tests, 1/4th the potency. Closely related to 2-aminotetralin.
2-Aminoindane - 2-AI(RC) Psychoactive compound. Rigid analogue of amphetamine.
5-(2-aminopropyl)indole - 5-IT(RC) indole derivative. Preparation was first reported in 1962 by Albert Hofmann. Positional isomer of AMT. Closer chemically resembles Phethylamines like 5-apb and the likes. Falls under the Analog act in the US with AMT.
6-(2-Aminopropyl)indole - ^. But it has been shown to increase hemoglobin levels in the bloodstream.
Aminorex - Known by many other names. Anorectic stimulant. Is classed within the 2-amino-5-aryl oxazoline class. Closely related to 4-methylaminorex. Shown to have locomotor stimulant effects, lying midway between dextro-amp and Meth. Attributed to the release of cathecholamines. Retired from the market after it was found to result in pulmonary hypertension.
2-Aminotetralin - (2-AT) consiting of a tetralin group combined with an anime. Rigid analogue of phenylisobutylamine. Fully substitutes for D-Amp in rat discrimination tests. Although at 1/8th the potency. Inhibits the reuptake of serotonin and norepinephrine. Likely induces their release as well. Also likely to act of Dopamine on account of the D-Amp.
Amiphenazole - Traditionally used as an antidote for Barb/opioid overdose. Mixed with bemegride. As well as poisoning from other depressants.
Ampyzine - Pyrazine derivative. That's all I could find with my limited research.
AR-R17779 - Drug that acts as a potent and selective full agonist for the α7 subtype of neural nicotinic acetylcholine receptors. Nootropic effects in animal sudies.
Armodafinal - Basically like all other versions of the ***final's nothing popped very interesting.
Bemegride - Used in barb overdoses. "Popularized" by The suspected Serial Killer Dr. John Bodkin Adams.
Benocyclidine - (BCP/BTCP) RC of the arylcyclohexylamine class. Acts as a Potent and Selective DRI. Pure DRI with negligible affintity for NMDA. Lacks every other propeties in effects, minus stimulant. Found in several MDMA presses.
3-benzhydrylmorpholine - Developed in the 50's by American Home Products Corp. Stimulant and anoretctic effects. Related to pipradrol and phenmetrazine.
Benzofuranylpropylaminopentance - ((-)-BPAP) Catecholaminergic and Serotonergic activity enhancer. Only increases the amount of neurotransmitters that get released. Weak MAO-A inhibitor. Showen to have neuroprotective effects similar to selegiling.
Benzooylthiomethylecgonine - Cocaine Analogue which has a sulfur in place of an oxygen on the single bonded benzoyl ester. Thus lowering potency.
1-Benzyl-4-(2-(diphenylmethoxy)ethyl)piperidine - Acts as a potent and selective DRI.
Benzylpipeazine - BZP, that's about it.
2-benzylpipeazine - 20x less potent than MPH and desoxypipadrol. Synthetic intermediate in other drugs :o. Boring stuff.
4-benzylpipeazine - The exact opposite of ^^. Acts as a MAOI with 20 to 48 fold selectivity for releasing dopamine versus serotonin.
Brasofensine - Phehyltropane. Effective in stimulating LMA and reversing akinesia. Idunknow.
Bromantane - Stimulant with anxiolytic properties developed in Russia during the late 1980's. DSRI. Has an anticholinergic effect at very high doses. Used as a doping agent for athletic performance. No withdrawal symptoms!
BTS 74,398 - Weird structure, centrally acting stimulant drug. Acts as a triple reuptake inhibitor.
Butylolylquinuclidine - Was made to replace cocaine in cocaine addiction, while longest lasting and less potent.
Camfetamine - N-Methyl homologue of fencamfamine. Apparently replaced mephedrone after it's banning?
Meta-Chlorophenylpiperazine
Cilboamine - NDRI, has stimulant and anti-dep effects.
Clofeniciclan - Dopamine-releasing agent developed in the 50's. Proved unpopular as a treatment because of its pronounced stimulant activity