Difference between revisions of "Quick Guide to Uncommon Stimulants"

Latest revision as of 03:18, 4 February 2014

2-MDP - Dissociative anaesthetic, NMDAN-methyl-D-aspartate receptor. NMDA antagonists are often dissociatives. antagonistA substance that interferes with or inhibits the physiological action of another., simlar effects to PCP in animals, (-) isomerEach of two or more compounds with the same formula but a different arrangement of atoms in the molecule and different properties. is active. Roughly 1/3rd potency of amphetamine by weight. Lasts over 24 hours.

2C-B-BZP - Benzylpiperazine base with ring-sub pattern of 2c-b. Not a phenethylaminePhenethylamine (PEA) is a natural monoamine alkaloid, trace amine, and psychoactive drug with stimulant effects. In the mammalian central nervous system, phenethylamine is believed to function as a neuromodulator or neurotransmitter., doesn't produce psychedelic effects. Lasts 3-6 hours. Was sold in Japan in "smartshops"

A-366/833 - AgonistA substance that initiates a physiological response when combined with a receptor. at neural nicotinic acetylcholine receptors selective for α4β2 subtype. Been researched as an analgesic. Hasn't passed clinical trials.

A-84/543 ^ That and is used as the "standard" for this family of compounds.

2-Acetoxycocaine - Quicker onset than Cocaine. Four fold increase over cocaine in binding potency for dopamineA neurotransmitter associated with movement, attention, learning, and the brain’s pleasure and reward system.. And 35 fold enhanced affinity for the norepinephrine. Reduced selectivity for serotoninA monoamine neurotransmitter, biochemically derived from tryptophan, that is primarily found in the gastrointestinal (GI) tract, platelets, and central nervous system (CNS) of humans and animals. It is a well-known contributor to feelings of well-being.. Interesting structure.

Adrafinil - Prodrug of Modafinil, unregulated in the US. 1 hour half life.

AL-1095 - Centrally acting, comparable effects to amp. developed by Bristol in the 70's.

Altinicline (SIB-1508Y) agonistA substance that initiates a physiological response when combined with a receptor. at neural nicotinic acetylcholine receptors similar to A-366. Releases DopamineA neurotransmitter associated with movement, attention, learning, and the brain’s pleasure and reward system. and Acetylcholine in both rodent and primate models. Progressed into Phase 2 clinical trials for Parkinson's.

Amfepramone - Diethylcathinone. By itself lacks any affinity for monoamine transporters and functions as a prodrug to ethcathinone. Very weak dopaminergic and serotonergic. 10-20x stronger on norepinephrine in comparison. Basically can be considered NRA's. Is currently Schedule IV in the United States. Class C drug in the UK. Apparently known as "tombstones" in the UK.

2-amino-1,2-dihydronaphthalene - Also known as 2-AD, rigid analogue of phenylisobutylamine and substitutes amphetamine for it in rat discrimination tests, 1/4th the potency. Closely related to 2-aminotetralin.

2-Aminoindane - 2-AI(RC) Psychoactive compound. Rigid analogue of amphetamine.

5-(2-aminopropyl)indole - 5-IT(RC) indole derivative. Preparation was first reported in 1962 by Albert Hofmann. Positional isomerEach of two or more compounds with the same formula but a different arrangement of atoms in the molecule and different properties. of AMT. Closer chemically resembles Phethylamines like 5-apb and the likes. Falls under the Analog act in the US with AMT.

6-(2-Aminopropyl)indole - ^. But it has been shown to increase hemoglobin levels in the bloodstream.

Aminorex - Known by many other names. Anorectic stimulant. Is classed within the 2-amino-5-aryl oxazoline class. Closely related to 4-methylaminorex. Shown to have locomotor stimulant effects, lying midway between dextro-amp and Meth. Attributed to the release of cathecholamines. Retired from the market after it was found to result in pulmonary hypertension.

2-Aminotetralin - (2-AT) consiting of a tetralin group combined with an anime. Rigid analogue of phenylisobutylamine. Fully substitutes for D-Amp in rat discrimination tests. Although at 1/8th the potency. Inhibits the reuptake of serotoninA monoamine neurotransmitter, biochemically derived from tryptophan, that is primarily found in the gastrointestinal (GI) tract, platelets, and central nervous system (CNS) of humans and animals. It is a well-known contributor to feelings of well-being. and norepinephrine. Likely induces their release as well. Also likely to act of DopamineA neurotransmitter associated with movement, attention, learning, and the brain’s pleasure and reward system. on account of the D-Amp.

Amiphenazole - Traditionally used as an antidote for Barb/opioid overdose. Mixed with bemegride. As well as poisoning from other depressants.

Ampyzine - Pyrazine derivative. That's all I could find with my limited research.

AR-R17779 - Drug that acts as a potent and selective full agonistA substance that initiates a physiological response when combined with a receptor. for the α7 subtype of neural nicotinic acetylcholine receptors. NootropicNootropics, also referred to as smart drugs, memory enhancers, neuro enhancers, cognitive enhancers, and intelligence enhancers, are drugs, supplements, nutraceuticals, and functional foods that purportedly improve mental functions such as cognition, memory, intelligence, motivation, attention, and concentration. They are generally neuroprotective, and non-toxic. effects in animal sudies.

Armodafinal - Basically like all other versions of the ***final's nothing popped very interesting.

Bemegride - Used in barb overdoses. "Popularized" by The suspected Serial Killer Dr. John Bodkin Adams.

Benocyclidine - (BCP/BTCP) RC of the arylcyclohexylamineA class of dissociatives, which includes PCP, Ketamine, Methoxetamine and others. An arylcyclohexylamine is composed of a cyclohexylamine unit with an aryl moiety attachment. The aryl group is positioned geminal to the amine. In the simplest cases, the aryl moiety is typically a phenyl ring, sometimes with additional substitution. The amine is usually not primary, secondary amines such as methylamino or ethylamino, or tertiary cycloalkylamines such as piperidino and pyrrolidino, are the most commonly encountered N-substituents. class. Acts as a Potent and Selective DRIDopamine Reuptake Inhibitor. Pure DRIDopamine Reuptake Inhibitor with negligible affintity for NMDAN-methyl-D-aspartate receptor. NMDA antagonists are often dissociatives.. Lacks every other propeties in effects, minus stimulant. Found in several MDMA presses.

3-benzhydrylmorpholine - Developed in the 50's by American Home Products Corp. Stimulant and anoretctic effects. Related to pipradrol and phenmetrazine.

Benzofuranylpropylaminopentance - ((-)-BPAP) Catecholaminergic and Serotonergic activity enhancer. Only increases the amount of neurotransmitters that get released. Weak MAOMonoamine Oxidase, an enzyme that catalyses the metabolism of many drugs (e.g., DMT, dopamine and serotonin).-A inhibitor. Showen to have neuroprotective effects similar to selegiling.

Benzooylthiomethylecgonine - Cocaine Analogue which has a sulfur in place of an oxygen on the single bonded benzoyl ester. Thus lowering potency.

1-Benzyl-4-(2-(diphenylmethoxy)ethyl)piperidine - Acts as a potent and selective DRIDopamine Reuptake Inhibitor.

Benzylpipeazine - BZP, that's about it.

2-benzylpipeazine - 20x less potent than MPH and desoxypipadrol. Synthetic intermediate in other drugs :o. Boring stuff.

4-benzylpipeazine - The exact opposite of ^^. Acts as a MAOIMonoamine oxidase inhibitor are drugs that inhibit the action of monoamine oxidase in the brain and so allow monoamines to accumulate. with 20 to 48 fold selectivity for releasing dopamineA neurotransmitter associated with movement, attention, learning, and the brain’s pleasure and reward system. versus serotoninA monoamine neurotransmitter, biochemically derived from tryptophan, that is primarily found in the gastrointestinal (GI) tract, platelets, and central nervous system (CNS) of humans and animals. It is a well-known contributor to feelings of well-being..

Brasofensine - Phehyltropane. Effective in stimulating LMA and reversing akinesia. Idunknow.

Bromantane - Stimulant with anxiolytic properties developed in Russia during the late 1980's. DSRI. Has an anticholinergic effect at very high doses. Used as a doping agent for athletic performance. No withdrawal symptoms!

BTS 74,398 - Weird structure, centrally acting stimulant drug. Acts as a triple reuptake inhibitor.

Butylolylquinuclidine - Was made to replace cocaine in cocaine addiction, while longest lasting and less potent.

Camfetamine - N-Methyl homologue of fencamfamine. Apparently replaced mephedrone after it's banning?

Meta-Chlorophenylpiperazine

Cilboamine - NDRINorepinephrine-Dopamine Reuptake Inhibitor, has stimulant and anti-dep effects.

Clofeniciclan - DopamineA neurotransmitter associated with movement, attention, learning, and the brain’s pleasure and reward system.-releasing agent developed in the 50's. Proved unpopular as a treatment because of its pronounced stimulant activity

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