Quick Guide to Uncommon Stimulants - Revision history

Sleep at 03:18, 4 February 2014

2014-02-04T03:18:19Z

← Older revision		Revision as of 22:18, 3 February 2014
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	:3-benzhydrylmorpholine - Developed in the 50's by American Home Products Corp. Stimulant and anoretctic effects. Related to pipradrol and phenmetrazine.		:3-benzhydrylmorpholine - Developed in the 50's by American Home Products Corp. Stimulant and anoretctic effects. Related to pipradrol and phenmetrazine.

			:Benzofuranylpropylaminopentance - ((-)-BPAP) Catecholaminergic and Serotonergic activity enhancer. Only increases the amount of neurotransmitters that get released. Weak MAO-A inhibitor. Showen to have neuroprotective effects similar to selegiling.

			:Benzooylthiomethylecgonine - Cocaine Analogue which has a sulfur in place of an oxygen on the single bonded benzoyl ester. Thus lowering potency.

			:1-Benzyl-4-(2-(diphenylmethoxy)ethyl)piperidine - Acts as a potent and selective DRI.

			:Benzylpipeazine - BZP, that's about it.

			:2-benzylpipeazine - 20x less potent than MPH and desoxypipadrol. Synthetic intermediate in other drugs :o. Boring stuff.

			:4-benzylpipeazine - The exact opposite of ^^. Acts as a MAOI with 20 to 48 fold selectivity for releasing dopamine versus serotonin.

			:Brasofensine - Phehyltropane. Effective in stimulating LMA and reversing akinesia. Idunknow.

			:Bromantane - Stimulant with anxiolytic properties developed in Russia during the late 1980's. DSRI. Has an anticholinergic effect at very high doses. Used as a doping agent for athletic performance. No withdrawal symptoms!

			:BTS 74,398 - Weird structure, centrally acting stimulant drug. Acts as a triple reuptake inhibitor.

			:Butylolylquinuclidine - Was made to replace cocaine in cocaine addiction, while longest lasting and less potent.

			:Camfetamine - N-Methyl homologue of fencamfamine. Apparently replaced mephedrone after it's banning?

			:Meta-Chlorophenylpiperazine

			:Cilboamine - NDRI, has stimulant and anti-dep effects.

			:Clofeniciclan - Dopamine-releasing agent developed in the 50's. Proved unpopular as a treatment because of its pronounced stimulant activity

Sleep at 16:32, 31 October 2013

2013-10-31T16:32:24Z

← Older revision		Revision as of 11:32, 31 October 2013
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	2-MDP - Dissociative anaesthetic, NMDA antagonist, simlar effects to PCP in animals, (-) isomer is active. Roughly 1/3rd potency of amphetamine by weight. Lasts over 24 hours.		:2-MDP - Dissociative anaesthetic, NMDA antagonist, simlar effects to PCP in animals, (-) isomer is active. Roughly 1/3rd potency of amphetamine by weight. Lasts over 24 hours.

	2C-B-BZP - Benzylpiperazine base with ring-sub pattern of 2c-b. Not a phenethylamine, doesn't produce psychedelic effects. Lasts 3-6 hours. Was sold in Japan in "smartshops"		:2C-B-BZP - Benzylpiperazine base with ring-sub pattern of 2c-b. Not a phenethylamine, doesn't produce psychedelic effects. Lasts 3-6 hours. Was sold in Japan in "smartshops"

	A-366/833 - Agonist at neural nicotinic acetylcholine receptors selective for α4β2 subtype. Been researched as an analgesic. Hasn't passed clinical trials.		:A-366/833 - Agonist at neural nicotinic acetylcholine receptors selective for α4β2 subtype. Been researched as an analgesic. Hasn't passed clinical trials.

	A-84/543 ^ That and is used as the "standard" for this family of compounds.		:A-84/543 ^ That and is used as the "standard" for this family of compounds.

	2-Acetoxycocaine - Quicker onset than Cocaine. Four fold increase over cocaine in binding potency for dopamine. And 35 fold enhanced affinity for the norepinephrine. Reduced selectivity for serotonin. Interesting structure.		:2-Acetoxycocaine - Quicker onset than Cocaine. Four fold increase over cocaine in binding potency for dopamine. And 35 fold enhanced affinity for the norepinephrine. Reduced selectivity for serotonin. Interesting structure.

	Adrafinil - Prodrug of Modafinil, unregulated in the US. 1 hour half life.		:Adrafinil - Prodrug of Modafinil, unregulated in the US. 1 hour half life.

	AL-1095 - Centrally acting, comparable ~~efffects~~ to amp. developed by Bristol in the 70's.		:AL-1095 - Centrally acting, comparable effects to amp. developed by Bristol in the 70's.

	Altinicline (SIB-1508Y) agonist at neural nicotinic acetylcholine receptors similar to A-366. Releases Dopamine and Acetylcholine in both rodent and primate models. Progressed into Phase 2 clinical trials for Parkinson's.		:Altinicline (SIB-1508Y) agonist at neural nicotinic acetylcholine receptors similar to A-366. Releases Dopamine and Acetylcholine in both rodent and primate models. Progressed into Phase 2 clinical trials for Parkinson's.

	Amfepramone - Diethylcathinone. By itself lacks any affinity for monoamine transporters and functions as a prodrug to ethcathinone. Very weak dopaminergic and serotonergic. 10-20x stronger on norepinephrine in comparison. Basically can be		:Amfepramone - Diethylcathinone. By itself lacks any affinity for monoamine transporters and functions as a prodrug to ethcathinone. Very weak dopaminergic and serotonergic. 10-20x stronger on norepinephrine in comparison. Basically can be considered NRA's. Is currently Schedule IV in the United States. Class C drug in the UK. Apparently known as "tombstones" in the UK.

	~~considered NRA's. Is currently Schedule IV in the United States. Class C drug in the UK. Apparently~~ known as ~~"tombstones"~~ in the UK.		:2-amino-1,2-dihydronaphthalene - Also known as 2-AD, rigid analogue of phenylisobutylamine and substitutes amphetamine for it in rat discrimination tests, 1/4th the potency. Closely related to 2-aminotetralin.

	2-~~amino~~-1,2-~~dihydronaphthalene - Also known as 2-AD, rigid~~ analogue of ~~phenylisobutylamine and substitutes~~ amphetamine ~~for it in rat discrimination tests, 1/4th the potency. Closely related to 2-aminotetralin~~.		:2-Aminoindane - 2-AI(RC) Psychoactive compound. Rigid analogue of amphetamine.

	2-~~Aminoindane~~ - 2-AI(RC) ~~Psychoactive compound~~. ~~Rigid analogue~~ of ~~amphetamine~~.		:5-(2-aminopropyl)indole - 5-IT(RC) indole derivative. Preparation was first reported in 1962 by Albert Hofmann. Positional isomer of AMT. Closer chemically resembles Phethylamines like 5-apb and the likes. Falls under the Analog act in the US with AMT.

	5-(2-~~aminopropyl~~)indole - ~~5-IT(RC) indole derivative~~. ~~Preparation was first reported~~ in ~~1962 by Albert Hofmann~~. ~~Positional isomer~~		:6-(2-Aminopropyl)indole - ^. But it has been shown to increase hemoglobin levels in the bloodstream.

	~~of AMT~~. ~~Closer chemically resembles Phethylamines like~~ 5-~~apb~~ and the ~~likes~~. ~~Falls under~~ the ~~Analog act~~ in ~~the US with AMT~~.		:Aminorex - Known by many other names. Anorectic stimulant. Is classed within the 2-amino-5-aryl oxazoline class. Closely related to 4-methylaminorex. Shown to have locomotor stimulant effects, lying midway between dextro-amp and Meth. Attributed to the release of cathecholamines. Retired from the market after it was found to result in pulmonary hypertension.

	6-(2-~~Aminopropyl~~)~~indole~~ - ^. ~~But it has been shown~~ to ~~increase hemoglobin levels in~~ the ~~bloodstream~~.		:2-Aminotetralin - (2-AT) consiting of a tetralin group combined with an anime. Rigid analogue of phenylisobutylamine. Fully substitutes for D-Amp in rat discrimination tests. Although at 1/8th the potency. Inhibits the reuptake of serotonin and norepinephrine. Likely induces their release as well. Also likely to act of Dopamine on account of the D-Amp.

	~~Aminorex~~ - ~~Known by many other names~~. ~~Anorectic stimulant~~. ~~Is classed within the 2-amino-5-aryl oxazoline class~~. ~~Closely related~~		:Amiphenazole - Traditionally used as an antidote for Barb/opioid overdose. Mixed with bemegride. As well as poisoning from other depressants.

	~~to 4~~-~~methylaminorex~~. ~~Shown to have locomotor stimulant effects, lying midway between dextro-amp and Meth~~. ~~Attributed to the~~		:Ampyzine - Pyrazine derivative. That's all I could find with my limited research.

	~~release~~ of ~~cathecholamines~~. ~~Retired from the market after it was found to result~~ in ~~pulmonary hypertension~~.		:AR-R17779 - Drug that acts as a potent and selective full agonist for the α7 subtype of neural nicotinic acetylcholine receptors. Nootropic effects in animal sudies.

	2-~~Aminotetralin - (2-AT) consiting of a tetralin group combined with an anime. Rigid analogue~~ of ~~phenylisobutylamine~~. ~~Fully~~		:Armodafinal - Basically like all other versions of the ***final's nothing popped very interesting.

	~~substitutes for D~~-~~Amp~~ in ~~rat discrimination tests~~. ~~Although at 1/8th the potenct~~. ~~Inhibits the reuptake of serotonin and~~		:Bemegride - Used in barb overdoses. "Popularized" by The suspected Serial Killer Dr. John Bodkin Adams.

	~~norepinephrine~~. ~~Likely induces their release~~ as ~~well~~. ~~Also likely to act of Dopamine on account of the D-Amp~~.		:Benocyclidine - (BCP/BTCP) RC of the arylcyclohexylamine class. Acts as a Potent and Selective DRI. Pure DRI with negligible affintity for NMDA. Lacks every other propeties in effects, minus stimulant. Found in several MDMA presses.

	~~Amiphenazole - Traditionally used as an antidote for Barb/opioid overdose. Mixed with bemegride. As well as poisoning from other depressants.~~		:3-benzhydrylmorpholine - Developed in the 50's by American Home Products Corp. Stimulant and anoretctic effects. Related to pipradrol and phenmetrazine.

	~~Ampyzine - Pyrazine derivative. That's all I could find with my limited research.~~

	~~AR-R17779 - Drug that acts as a potent and selective full agonist for the α7 subtype of neural nicotinic acetylcholine receptors. Nootropic effects in animal sudies.~~

	~~Armodafinal - Basically like all other versions of the ***final's nothing popped very interesting.~~

	~~Bemegride - Used in barb overdoses. "Popularized" by The suspected Serial Killer Dr. John Bodkin Adams.~~

	~~Benocyclidine - (BCP/BTCP) RC of the arylcyclohexylamine class. Acts as a Potent and Selective DRI. Pure DRI with negligible~~

	~~affintity for NMDA. Lacks every other propeties in effects, minus stimulant. Found in several MDMA presses.~~

	3-benzhydrylmorpholine - Developed in the 50's by American Home Products Corp. Stimulant and anoretctic effects. Related to pipradrol and phenmetrazine.

Sleep at 05:42, 20 September 2013

2013-09-20T05:42:10Z

← Older revision		Revision as of 00:42, 20 September 2013
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	Altinicline (SIB-1508Y) agonist at neural nicotinic acetylcholine receptors similar to A-366. Releases Dopamine and Acetylcholine in both rodent and primate models. Progressed into Phase 2 clinical trials for Parkinson's.		Altinicline (SIB-1508Y) agonist at neural nicotinic acetylcholine receptors similar to A-366. Releases Dopamine and Acetylcholine in both rodent and primate models. Progressed into Phase 2 clinical trials for Parkinson's.

	Amfepramone - Diethylcathinone. By itself lacks any affinity for monoamine transporters and functions as a prodrug to ethcathinone. Very weak dopaminergic and serotonergic. 10-20x stronger on norepinephrine in comparison. Basically can be considered NRA's. Is currently Schedule IV in the United States. Class C drug in the UK. Apparently known as "tombstones" in the UK.		Amfepramone - Diethylcathinone. By itself lacks any affinity for monoamine transporters and functions as a prodrug to ethcathinone. Very weak dopaminergic and serotonergic. 10-20x stronger on norepinephrine in comparison. Basically can be

			considered NRA's. Is currently Schedule IV in the United States. Class C drug in the UK. Apparently known as "tombstones" in the UK.

	2-amino-1,2-dihydronaphthalene - Also known as 2-AD, rigid analogue of phenylisobutylamine and substitutes amphetamine for it in rat discrimination tests, 1/4th the potency. Closely related to 2-aminotetralin.		2-amino-1,2-dihydronaphthalene - Also known as 2-AD, rigid analogue of phenylisobutylamine and substitutes amphetamine for it in rat discrimination tests, 1/4th the potency. Closely related to 2-aminotetralin.
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	2-Aminoindane - 2-AI(RC) Psychoactive compound. Rigid analogue of amphetamine.		2-Aminoindane - 2-AI(RC) Psychoactive compound. Rigid analogue of amphetamine.

	5-(2-aminopropyl)indole - 5-IT(RC) indole derivative. Preparation was first reported in 1962 by Albert Hofmann. Positional isomer ~~of AMT. Closer chemically resembles~~		5-(2-aminopropyl)indole - 5-IT(RC) indole derivative. Preparation was first reported in 1962 by Albert Hofmann. Positional isomer

	Phethylamines like 5-apb and the likes. Falls under the Analog act in the US with AMT.		of AMT. Closer chemically resembles Phethylamines like 5-apb and the likes. Falls under the Analog act in the US with AMT.

	6-(2-Aminopropyl)indole - ^. But it has been shown to increase hemoglobin levels in the bloodstream.		6-(2-Aminopropyl)indole - ^. But it has been shown to increase hemoglobin levels in the bloodstream.

	Aminorex - Known by many other names. Anorectic stimulant. Is classed within the 2-amino-5-aryl oxazoline class. Closely related to 4-methylaminorex. Shown to have locomotor stimulant effects, lying midway between dextro-amp and Meth. Attributed to the release of cathecholamines. Retired from the market after it was found to result in pulmonary hypertension.		Aminorex - Known by many other names. Anorectic stimulant. Is classed within the 2-amino-5-aryl oxazoline class. Closely related

			to 4-methylaminorex. Shown to have locomotor stimulant effects, lying midway between dextro-amp and Meth. Attributed to the

			release of cathecholamines. Retired from the market after it was found to result in pulmonary hypertension.

			2-Aminotetralin - (2-AT) consiting of a tetralin group combined with an anime. Rigid analogue of phenylisobutylamine. Fully

			substitutes for D-Amp in rat discrimination tests. Although at 1/8th the potenct. Inhibits the reuptake of serotonin and

			norepinephrine. Likely induces their release as well. Also likely to act of Dopamine on account of the D-Amp.

			Amiphenazole - Traditionally used as an antidote for Barb/opioid overdose. Mixed with bemegride. As well as poisoning from other depressants.

			Ampyzine - Pyrazine derivative. That's all I could find with my limited research.

			AR-R17779 - Drug that acts as a potent and selective full agonist for the α7 subtype of neural nicotinic acetylcholine receptors. Nootropic effects in animal sudies.

			Armodafinal - Basically like all other versions of the ***final's nothing popped very interesting.

			Bemegride - Used in barb overdoses. "Popularized" by The suspected Serial Killer Dr. John Bodkin Adams.

			Benocyclidine - (BCP/BTCP) RC of the arylcyclohexylamine class. Acts as a Potent and Selective DRI. Pure DRI with negligible

	~~2-Aminotetralin - (2-AT) consiting of a tetralin group combined with an anime~~. ~~Rigid analogue of phenylisobutylamine~~. ~~Fully substitutes for D-Amp~~ in ~~rat discrimination tests~~.		affintity for NMDA. Lacks every other propeties in effects, minus stimulant. Found in several MDMA presses.

	~~Although at 1/8th~~ the ~~potenct~~. ~~Inhibits the reuptake of serotonin~~ and ~~norepinephrine~~. ~~Likely induces their release as well. Also likely~~ to ~~act of Dopamine on account of the D-Amp~~.		3-benzhydrylmorpholine - Developed in the 50's by American Home Products Corp. Stimulant and anoretctic effects. Related to pipradrol and phenmetrazine.

Sleep at 02:34, 19 September 2013

2013-09-19T02:34:59Z

← Older revision		Revision as of 21:34, 18 September 2013
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	2-MDP - Dissociative anaesthetic, NMDA antagonist, simlar effects to PCP in animals, (-) isomer is active. Roughly 1/3rd		2-MDP - Dissociative anaesthetic, NMDA antagonist, simlar effects to PCP in animals, (-) isomer is active. Roughly 1/3rd potency of amphetamine by weight. Lasts over 24 hours.

	~~potency~~ of ~~amphetamine by weight~~. Lasts ~~over 24~~ hours.		2C-B-BZP - Benzylpiperazine base with ring-sub pattern of 2c-b. Not a phenethylamine, doesn't produce psychedelic effects. Lasts 3-6 hours. Was sold in Japan in "smartshops"

	2C-B-~~BZP - Benzylpiperazine base with ring-sub pattern of 2c-b~~. ~~Not a phenethylamine, doesn~~'t ~~produce psychedelic effects~~.		A-366/833 - Agonist at neural nicotinic acetylcholine receptors selective for α4β2 subtype. Been researched as an analgesic. Hasn't passed clinical trials.

	~~Lasts 3~~-~~6 hours. Was sold in Japan in~~ "~~smartshops~~"		A-84/543 ^ That and is used as the "standard" for this family of compounds.

	A-~~366/833~~ - ~~Agonist at neural nicotinic acetylcholine receptors selective~~ for ~~α4β2 subtype~~. ~~Been researched as an analgesic~~.		2-Acetoxycocaine - Quicker onset than Cocaine. Four fold increase over cocaine in binding potency for dopamine. And 35 fold enhanced affinity for the norepinephrine. Reduced selectivity for serotonin. Interesting structure.

	~~Hasn't passed clinical trials~~.		Adrafinil - Prodrug of Modafinil, unregulated in the US. 1 hour half life.

	A-~~84/543 ^ That~~ and ~~is used~~ as the "~~standard~~" for ~~this family of compounds~~.		AL-1095 - Centrally acting, comparable efffects to amp. developed by Bristol in the 70's.

			Altinicline (SIB-1508Y) agonist at neural nicotinic acetylcholine receptors similar to A-366. Releases Dopamine and Acetylcholine in both rodent and primate models. Progressed into Phase 2 clinical trials for Parkinson's.

			Amfepramone - Diethylcathinone. By itself lacks any affinity for monoamine transporters and functions as a prodrug to ethcathinone. Very weak dopaminergic and serotonergic. 10-20x stronger on norepinephrine in comparison. Basically can be considered NRA's. Is currently Schedule IV in the United States. Class C drug in the UK. Apparently known as "tombstones" in the UK.

			2-amino-1,2-dihydronaphthalene - Also known as 2-AD, rigid analogue of phenylisobutylamine and substitutes amphetamine for it in rat discrimination tests, 1/4th the potency. Closely related to 2-aminotetralin.

	2-~~Acetoxycocaine~~ - ~~Quicker onset than Cocaine~~. ~~Four fold increase over cocaine in binding potency for dopamine~~. ~~And 35 fold~~		2-Aminoindane - 2-AI(RC) Psychoactive compound. Rigid analogue of amphetamine.

	~~enhanced affinity for the norepinephrine~~. ~~Reduced selectivity for serotonin~~. ~~Interesting structure~~.		5-(2-aminopropyl)indole - 5-IT(RC) indole derivative. Preparation was first reported in 1962 by Albert Hofmann. Positional isomer of AMT. Closer chemically resembles

	~~Adrafinil~~ - ~~Prodrug of Modafinil, unregulated~~ in the US~~. 1 hour half life~~.		Phethylamines like 5-apb and the likes. Falls under the Analog act in the US with AMT.

	AL-~~1095~~ - ~~Centrally acting, comparable efffects~~ to ~~amp. developed by Bristol~~ in the ~~70's~~.		6-(2-Aminopropyl)indole - ^. But it has been shown to increase hemoglobin levels in the bloodstream.

	~~Altinicline (SIB~~-~~1508Y) agonist at neural nicotinic acetylcholine receptors similar~~ to A-~~366~~. ~~Releases Dopamine~~ and		Aminorex - Known by many other names. Anorectic stimulant. Is classed within the 2-amino-5-aryl oxazoline class. Closely related to 4-methylaminorex. Shown to have locomotor stimulant effects, lying midway between dextro-amp and Meth. Attributed to the release of cathecholamines. Retired from the market after it was found to result in pulmonary hypertension.

	~~Acetylcholine in both rodent and primate models~~. ~~Progressed into Phase 2 clinical trials~~ for ~~Parkinson's~~.		2-Aminotetralin - (2-AT) consiting of a tetralin group combined with an anime. Rigid analogue of phenylisobutylamine. Fully substitutes for D-Amp in rat discrimination tests.

	~~Amfepramone - Diethylcathinone~~. ~~By itself lacks any affinity for monoamine transporters~~ and ~~functions~~ as ~~a prodrug~~ to ~~ethcathinone. Very weak dopaminergic and serotonergic. 10-20x stronger~~ on ~~norepinephrine in comparison. Basically can be considered NRA's. Is currently Schedule IV in~~ the ~~United States. Class C drug in the UK. Apparently known as "tombstones" in the UK~~.		Although at 1/8th the potenct. Inhibits the reuptake of serotonin and norepinephrine. Likely induces their release as well. Also likely to act of Dopamine on account of the D-Amp.

Sleep: Created page with "2-MDP - Dissociative anaesthetic, NMDA antagonist, simlar effects to PCP in animals, (-) isomer is active. Roughly 1/3rd potency of amphetamine by weight. Lasts over 24 hour..."

2013-09-19T01:31:03Z

Created page with "2-MDP - Dissociative anaesthetic, NMDA antagonist, simlar effects to PCP in animals, (-) isomer is active. Roughly 1/3rd potency of amphetamine by weight. Lasts over 24 hour..."

New page

2-MDP - Dissociative anaesthetic, NMDA antagonist, simlar effects to PCP in animals, (-) isomer is active. Roughly 1/3rd

potency of amphetamine by weight. Lasts over 24 hours.

2C-B-BZP - Benzylpiperazine base with ring-sub pattern of 2c-b. Not a phenethylamine, doesn't produce psychedelic effects.

Lasts 3-6 hours. Was sold in Japan in "smartshops"

A-366/833 - Agonist at neural nicotinic acetylcholine receptors selective for α4β2 subtype. Been researched as an analgesic.

Hasn't passed clinical trials.

A-84/543 ^ That and is used as the "standard" for this family of compounds.

2-Acetoxycocaine - Quicker onset than Cocaine. Four fold increase over cocaine in binding potency for dopamine. And 35 fold

enhanced affinity for the norepinephrine. Reduced selectivity for serotonin. Interesting structure.

Adrafinil - Prodrug of Modafinil, unregulated in the US. 1 hour half life.

AL-1095 - Centrally acting, comparable efffects to amp. developed by Bristol in the 70's.

Altinicline (SIB-1508Y) agonist at neural nicotinic acetylcholine receptors similar to A-366. Releases Dopamine and

Acetylcholine in both rodent and primate models. Progressed into Phase 2 clinical trials for Parkinson's.

Amfepramone - Diethylcathinone. By itself lacks any affinity for monoamine transporters and functions as a prodrug to ethcathinone. Very weak dopaminergic and serotonergic. 10-20x stronger on norepinephrine in comparison. Basically can be considered NRA's. Is currently Schedule IV in the United States. Class C drug in the UK. Apparently known as "tombstones" in the UK.